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Ethionamide boosters. 2. Combining bioisosteric replacement and structure-based drug design to solve pharmacokinetic issues in a series of potent 1,2,4-oxadiazole EthR inhibitors31058
Publication Type: Peer reviewed scientific article Authors: Flipo,M.; Desroses,M.; Lecat-Guillet,N.; Villemagne,B.; Blondiaux,N.; Leroux,F.; Piveteau,C.; Vanessa Mathys; Flament,M.P.; Siepmann,J.; ...
Reversion of antibiotic resistance in Mycobacterium tuberculosis by spiroisoxazoline SMARt-420.
Publication Type: Peer reviewed scientific article Authors: Blondiaux, Nicolas; Moune, Martin; Desroses, Matthieu; Frita, Rosangela; Flipo, Marion; Vanessa Mathys; Karine Soetaert; Kiass, Mehdi; ...
The small-molecule SMARt751 reverses resistance to ethionamide in acute and chronic mouse models of tuberculosis.
Publication Type: Peer reviewed scientific article Authors: Flipo, Marion; Frita, Rosangela; Marilyne Bourotte; Maria S Martínez-Martínez; Markus Boesche; Gary W Boyle; Geo Derimanov; Gerard Drewes; ...