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Ethionamide boosters. 2. Combining bioisosteric replacement and structure-based drug design to solve pharmacokinetic issues in a series of potent 1,2,4-oxadiazole EthR inhibitors31058
Publication Type: Peer reviewed scientific article Authors: Flipo,M.; Desroses,M.; Lecat-Guillet,N.; Villemagne,B.; Blondiaux,N.; Leroux,F.; Piveteau,C.; Vanessa Mathys; Flament,M.P.; Siepmann,J.; ...
The small-molecule SMARt751 reverses resistance to ethionamide in acute and chronic mouse models of tuberculosis.
Piveteau; Kiass, Mehdi; Vanessa Mathys; Karine Soetaert; Véronique Megalizzi; Tanina, Abdalkarim; Wintjens, René; Antoine, Rudy; Brodin, Priscille; Delorme, Vincent; Moune, Martin; Djaout, Kamel; Stéphanie ...