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Ethionamide boosters. 2. Combining bioisosteric replacement and structure-based drug design to solve pharmacokinetic issues in a series of potent 1,2,4-oxadiazole EthR inhibitors31058
Models,Molecular Mycobacterium Mycobacterium tuberculosis ON Oxadiazoles pathogen Pharmacokinetic pharmacokinetics Piperidines PROCESSES Prodrugs protein Proteins Repressor Proteins Research Research Support SB- IM ...
Synthesis and biological activity of endomorphin-2 analogs incorporating piperidine-2-, 3- or 4-carboxylic acids instead of proline in position 24391
chemistry Comparison electronic Functional im Inhibitory Concentration 50 Institute IS journal Laboratories medical Oligopeptides Piperidines Proline rats Receptor receptors Receptors,Opioid,mu Research ...