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Résultats de la recherche - 12 results
RNA-based drug susceptibility testing of Mycobacterium tuberculosis
Publication Type: Scientific poster, presentation or proceeding Authors: An Van den Bossche; Roby Bhattacharyya; Jean-Yves Coppee; Leen Rigouts; Alain Baulard; Deborah Hung; Vanessa Mathys; ...
Ethionamide boosters. 2. Combining bioisosteric replacement and structure-based drug design to solve pharmacokinetic issues in a series of potent 1,2,4-oxadiazole EthR inhibitors31058
Villeret,V.; Wohlkonig,A.; Wintjens,R.; Soror,S.H.; Christophe,T.; Jeon,H.K.; Locht,C.; Brodin,P.; Deprez,B.; Baulard,A.R.; Willand,N. Source: J.Med.Chem., Volume 55, Issue 1, Number 83, p.68- 83 (2012) ...
Synthetic EthR inhibitors boost antituberculous activity of ethionamide36849
Delcroix,G.; Frenois,F.; Aumercier,M.; Locht,C.; Villeret,V.; Deprez,B.; Baulard,A.R. Source: Nat.Med., Volume 15, Issue 5, Number 544, p.537- 544 (2009) Keywords: 0 a Activity Agent Agents Animals antagonists ...
Molecular genetics of para-aminosalicylic acid resistance in clinical isolates and spontaneous mutants of Mycobacterium tuberculosis.
Mathema, Barun; Baulard, Alain; Kreiswirth, Barry N; Bifani, Pablo Source: Antimicrob Agents Chemother, Volume 53, Issue 5, p.2100-9 (2009) Keywords: Aminosalicylic Acid Antitubercular Agents Bacterial ...
The anti-cancer drug 5-fluorouracil is highly active against Mycobacterium tuberculosis in vitro but not in vivo
Publication Type: Scientific poster, presentation or proceeding Authors: Vanessa Mathys; Singhal,A.; Kiass,M.; P. Lefevre; Kurepina,N.; Wang,X.M.; Mathema,B.; Baulard,A.; Bifani,P. Source: ...
Mutations associated with para-aminosalicylic acid (PAS) resistance in clinical isolates and spontaneous mutants of Mycobacterium tuberculosis
Publication Type: Scientific poster, presentation or proceeding Authors: Vanessa Mathys; Quatannens,J.; Wintjens,R.; Kurepina,N.; Singhal,A.; Kiass,M.; Mathema,B.; Baulard,A.; B.N. Kreiswirth; ...
Molecular characterization of genes associated with ethionamide resistance in Mycobacterium tuberculosis clinical isolates and spontaneous mutants
Publication Type: Scientific poster, presentation or proceeding Authors: Vanessa Mathys; Baulard,A.; Kurepina,N.; M. Fauville; B.N. Kreiswirth; Bifani,P. Source: 106th General Meeting, NA, Issue ...
Mutations associated with PAS resistance in clinical isolates and spontaneous mutants of Mycobaterium tuberculosis
Publication Type: Scientific poster, presentation or proceeding Authors: Vanessa Mathys; Quatannens,J.; Kurepina,N.; Wintjens,R.; Mathema,B.; Baulard,A.; B.N. Kreiswirth; Bifani,P.; Belgian Society ...
Reversion of antibiotic resistance in Mycobacterium tuberculosis by spiroisoxazoline SMARt-420.
Locht, Camille; Brodin, Priscille; Gitzinger, Marc; Déprez, Benoit; Willand, Nicolas; Baulard, Alain R Source: Science, Volume 355, Issue 6330, p.1206-1211 (2017) Abstract: Antibiotic resistance is one of ...
RNA-based drug susceptibility testing of Mycobacterium tuberculosis
Publication Type: Scientific poster, presentation or proceeding Authors: An Van den Bossche; Roby Bhattacharyya; Jean-Yves Coppee; Leen Rigouts; Alain Baulard; Alexandra Vodolazkaia; Deborah Hung; ...