Search results - 16 results

In vitro and in vivo local tolerability of a synergistic anti-tuberculosis drug combination intended for pulmonary delivery.

Nathalie Source: J Appl Toxicol, Volume 43, Issue 2 (2023) Keywords: Alveolar Epithelial Cells Animals Antitubercular Agents Bronchoalveolar Lavage Fluid Humans Lung mice Mycobacterium tuberculosis Orlistat ...

Phytochemical and in vitro antimicrobial and genotoxic activity in the brown algae Dictyopteris membranacea

(2017) Keywords: Antimicrobial activity Antitubercular activity Dictyopteris membranacea Micronucleus test Phytochemical analysis Vitotox test Health Topics:  Health and environment Santé et environnement ...

External quality assessment for tuberculosis diagnosis and drug resistance in the European Union: A five year multicentre implementation study

Volume 11, Issue 4, p.e0152926 (2016) Keywords: 0 a accuracy Activity Agent Agents ALL Amikacin Antitubercular Agents Area article AS assessment Benefit benefits Clinical Laboratory Techniques Common ...

Synthesis and anti-tubercular activity of N(2)-arylbenzo[g]isoquinoline-5,10-dione-3-iminium bromides.

Abbaspour Tehrani, K Source: Org Biomol Chem, Volume 14, Issue 6, p.2041-51 (2016) Keywords: Antitubercular Agents Dose-Response Relationship, Drug Hydrocarbons, Brominated Isoquinolines Macrophages Microbial ...

Anti-mycobacterial activity of 1,3-diaryltriazenes.

Polanc, Slovenko; Huygen, Kris; Košmrlj, Janez Source: Eur J Med Chem, Volume 77, p.193-203 (2014) Keywords: Animals Antitubercular Agents Cell Line Cell Survival Dose-Response Relationship, Drug ...

2,4-Dialkyl-8,9,10,11-tetrahydrobenzo[g]pyrimido[4,5-c]isoquinoline-1,3,7,12(2H,4H)-tetraones as new leads against Mycobacterium tuberculosis.

Norbert Source: Eur J Med Chem, Volume 77, p.409-21 (2014) Keywords: Animals Antitubercular Agents Cell Line Dose-Response Relationship, Drug Isoquinolines Macrophages mice Microbial Sensitivity Tests ...

Biological evaluation of diazene derivatives as anti-tubercular compounds.

Huygen, Kris; Košmrlj, Janez Source: Eur J Med Chem, Volume 74, p.85-94 (2014) Keywords: Antitubercular Agents Drug Screening Assays, Antitumor Imides Abstract: Despite efforts made in chemotherapeutic ...

Para-Aminosalicylic acid is a prodrug targeting dihydrofolate reductase in Mycobacterium tuberculosis33991

J.Biol.Chem., Volume 288, Issue 32, Number 23456, p.23447- 23456 (2013) Keywords: 0 a acid Activity Agent Agents Aminosalicylic Acid an antagonists & inhibitors Antitubercular Agents article AS Bacterial ...

Biological evaluation of bisbenzaldehydes against four Mycobacterium species.

Vanden Eynde, Jean Jacques; Huygen, Kris Source: Eur J Med Chem, Volume 63, p.731-8 (2013) Keywords: Animals Anti-Bacterial Agents Antitubercular Agents Benzaldehydes Cell Line Cell Survival Cells, ...

Systematic analysis of pyrazinamide-resistant spontaneous mutants and clinical isolates of Mycobacterium tuberculosis.

is a first-line antitubercular drug known for its activity against persistent Mycobacterium tuberculosis bacilli. We set out to systematically determine the PZA susceptibility profiles and mutations in ...

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