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Novel highly potent mu-opioid receptor antagonist based on endomorphin-2 structure4392
Bioorg.Med.Chem.Lett., Volume 18, Issue 4, Number 1353, p.1350- 1353 (2008) Keywords: 0 a Activity Aequorin agonists an Analgesics Analgesics,Opioid Animals antagonists & inhibitors article AS Calcium chemical ...
Mu-opioid receptor ligands lack receptor subtype selectivity in the aequorin luminescence-based calcium assay4393
(2007) Keywords: 0 a Aequorin agonists ALL an analysis Animals antagonists & inhibitors article Calcium Cell cells Change Changes chemistry Cho Cells classification Cricetinae Cricetulus effect ...
Synthesis and characterization of potent and selective mu-opioid receptor antagonists, [Dmt(1), D-2-Nal(4)]endomorphin-1 (Antanal-1) and [Dmt(1), D-2-Nal(4)]endomorphin-2 (Antanal-2)4395
Volume 50, Issue 3, Number 520, p.512- 520 (2007) Keywords: 0 a Aequorin Agent Agents agonists Analgesics Animals antagonists & inhibitors article AS Binding Sites brain Calcium chemical synthesis ...
[D-1-Nal4]endomorphin-2 is a potent micro-opioid receptor antagonist in the aequorin luminescence-based calcium assay4398
1099, p.1094- 1099 (2006) Keywords: 0 a Aequorin agonists analysis Animals antagonists & inhibitors article Biological Assay Calcium Cell Cell Line Change Changes chemistry Cho Cells Cricetinae data ...
Comparison of antagonist activity of spantide family at human neurokinin receptors measured by aequorin luminescence-based functional calcium assay4401
Keywords: 0 a Activity Aequorin Agent Agents ALL Analgesics analogs & derivatives Animals antagonists & inhibitors article AS at Biological Assay Calcium Cell Cell Line Change Changes chemistry Cho ...