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Résultats de la recherche - 3 results
Ethionamide boosters. 2. Combining bioisosteric replacement and structure-based drug design to solve pharmacokinetic issues in a series of potent 1,2,4-oxadiazole EthR inhibitors31058
Publication Type: Peer reviewed scientific article Authors: Flipo,M.; Desroses,M.; Lecat-Guillet,N.; Villemagne,B.; Blondiaux,N.; Leroux,F.; Piveteau,C.; Vanessa Mathys; Flament,M.P.; Siepmann,J.; ...
Synthetic EthR inhibitors boost antituberculous activity of ethionamide36849
Publication Type: Peer reviewed scientific article Authors: Willand,N.; Dirie,B.; Carette,X.; Bifani,P.; Singhal,A.; Desroses,M.; Leroux,F.; Willery,E.; Vanessa Mathys; Deprez-Poulain,R.; ...
Reversion of antibiotic resistance in Mycobacterium tuberculosis by spiroisoxazoline SMARt-420.
Publication Type: Peer reviewed scientific article Authors: Blondiaux, Nicolas; Moune, Martin; Desroses, Matthieu; Frita, Rosangela; Flipo, Marion; Vanessa Mathys; Karine Soetaert; Kiass, Mehdi; ...