- Vouliez-vous dire
- willebrand,n.
Résultats de la recherche - 4 results
Ethionamide boosters. 2. Combining bioisosteric replacement and structure-based drug design to solve pharmacokinetic issues in a series of potent 1,2,4-oxadiazole EthR inhibitors31058
Villeret,V.; Wohlkonig,A.; Wintjens,R.; Soror,S.H.; Christophe,T.; Jeon,H.K.; Locht,C.; Brodin,P.; Deprez,B.; Baulard,A.R.; Willand,N. Source: J.Med.Chem., Volume 55, Issue 1, Number 83, p.68- 83 (2012) ...
Synthetic EthR inhibitors boost antituberculous activity of ethionamide36849
Publication Type: Peer reviewed scientific article Authors: Willand,N.; Dirie,B.; Carette,X.; Bifani,P.; Singhal,A.; Desroses,M.; Leroux,F.; Willery,E.; Vanessa Mathys; Deprez-Poulain,R.; ...
Reversion of antibiotic resistance in Mycobacterium tuberculosis by spiroisoxazoline SMARt-420.
Locht, Camille; Brodin, Priscille; Gitzinger, Marc; Déprez, Benoit; Willand, Nicolas; Baulard, Alain R Source: Science, Volume 355, Issue 6330, p.1206-1211 (2017) Abstract: Antibiotic resistance is one of ...
The small-molecule SMARt751 reverses resistance to ethionamide in acute and chronic mouse models of tuberculosis.
Slupek; Kemmer, Christian; Gitzinger, Marc; Lluis Ballell; Alfonso Mendoza-Losana; Sergio Lociuro; Déprez, Benoit; David Barros-Aguirre; Modesto J Remuiñán; Willand, Nicolas; Baulard, Alain R Source: Sci ...