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Synthetic EthR inhibitors boost antituberculous activity of ethionamide36849

Publication Type: Peer reviewed scientific article Authors: Willand,N.; Dirie,B.; Carette,X.; Bifani,P.; Singhal,A.; Desroses,M.; Leroux,F.; Willery,E.; Vanessa Mathys; Deprez-Poulain,R.; ...

Reversion of antibiotic resistance in Mycobacterium tuberculosis by spiroisoxazoline SMARt-420.

Locht, Camille; Brodin, Priscille; Gitzinger, Marc; Déprez, Benoit; Willand, Nicolas; Baulard, Alain R Source: Science, Volume 355, Issue 6330, p.1206-1211 (2017) Abstract: Antibiotic resistance is one of ...

The small-molecule SMARt751 reverses resistance to ethionamide in acute and chronic mouse models of tuberculosis.

Slupek; Kemmer, Christian; Gitzinger, Marc; Lluis Ballell; Alfonso Mendoza-Losana; Sergio Lociuro; Déprez, Benoit; David Barros-Aguirre; Modesto J Remuiñán; Willand, Nicolas; Baulard, Alain R Source: Sci ...

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