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Zoekresultaten - 12 results

Identification of endomorphin-1 and endomorphin-2 binding sites in human mu-opioid receptor by antisense oligonucleotide strategy4389

Number 512, p.507- 512 (2008) Keywords: 0 a Aequorin ALL Analgesics Analgesics,Opioid analysis Animals antagonists & inhibitors article AS at Base Sequence Binding Sites Calcium Cell cells chemistry ...

Synthesis and biological activity of endomorphin-2 analogs incorporating piperidine-2-, 3- or 4-carboxylic acids instead of proline in position 24391

Number 94, p.91- 94 (2008) Keywords: 0 acid Acids Activity Aequorin Amino Acid Substitution Amino acids an Animals antagonists & inhibitors article AS brain Brain Chemistry Calcium Carboxylic Acids ...

Novel highly potent mu-opioid receptor antagonist based on endomorphin-2 structure4392

Bioorg.Med.Chem.Lett., Volume 18, Issue 4, Number 1353, p.1350- 1353 (2008) Keywords: 0 a Activity Aequorin agonists an Analgesics Analgesics,Opioid Animals antagonists & inhibitors article AS Calcium chemical ...

Mu-opioid receptor ligands lack receptor subtype selectivity in the aequorin luminescence-based calcium assay4393

(2007) Keywords: 0 a Aequorin agonists ALL an analysis Animals antagonists & inhibitors article Calcium Cell cells Change Changes chemistry Cho Cells classification Cricetinae Cricetulus effect ...

Characterization of tachykinin-related peptides from different insect species on Drosophila tachykinin receptor-expressing cell line4396

agonist induces a transient increase in the concentration of intracellular calcium. The functional assay based on aequorin-derived luminescence triggered by receptor-mediated changes in Ca(2+) levels was ...

[D-1-Nal4]endomorphin-2 is a potent micro-opioid receptor antagonist in the aequorin luminescence-based calcium assay4398

1099, p.1094- 1099 (2006) Keywords: 0 a Aequorin agonists analysis Animals antagonists & inhibitors article Biological Assay Calcium Cell Cell Line Change Changes chemistry Cho Cells Cricetinae data ...

Functional characterization of opioid receptor ligands by aequorin luminescence-based calcium assay4399

Issue 3, Number 1154, p.1150- 1154 (2006) Keywords: 0 a Aequorin Agent Agents agonists Analgesics Analgesics,Opioid analysis Animal Animals application article AS at Biological Assay biosynthesis Calcium ...

Comparison of antagonist activity of spantide family at human neurokinin receptors measured by aequorin luminescence-based functional calcium assay4401

Keywords: 0 a Activity Aequorin Agent Agents ALL Analgesics analogs & derivatives Animals antagonists & inhibitors article AS at Biological Assay Calcium Cell Cell Line Change Changes chemistry Cho ...

Substitution of conserved glycine residue by alanine in natural and synthetic neuropeptide ligands causes partial agonism at the stomoxytachykinin receptor4407

Vanden Broeck Source: J.Neurochem., Volume 90, Issue 2, Number 478, p.472- 478 (2004) Keywords: 0 a Aequorin agonists Alanine Amino Acid Sequence Amino Acid Substitution an Animals Apoproteins article AS ...

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